Affinité et efficacité des agonistes partiels et complets non peptidiques du récepteur OTR.
| Composé Ferring | WAY-267464 | LIT-001 | |
|---|---|---|---|
| OTR affinité (Ki, nM) | 141 | 30,5 | 61 |
| OTR agonisme (EC50, nM) | 28 (84 % max.) | 24 (70 % max.) | 25 (96 %) |
| V1AR affinité (KI, nM) | 196 | 12,5 | 1253 |
| V1AR antagonisme (IC50, nM) | 8 | 7 | 100 |
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